CYP-450 inducers are –
Correct Answer: Phenobarbitone
Description: Ans. is 'c' i.e., Phenobarbitone Drugs that induce microsomal enzymes o Phenobarbitone o Rifampin o Isoniazid o Phenylbutazone o DDT o Carbamezepine o Clofibrate o Ritonavir o Chronic alcohol intake o Cyclophosphamide o Phenytoin o Glucocoicoids o Chloral hydrate o Griseofulvin o Omeprazole o Meprobamate o Glutethimide o Cigarette smoking Remember o All Barbiturates are enzyme inducers except secobarbital, which inhibits the enzyme. o Acutely, ritonavir is an inhibitor, while with chronic (repeated) administration it acts as an inducer.
Category:
Pharmacology
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